Potassium channel opener


A potassium channel opener is a type of drug which facilitates ion transmission through potassium channels.

Examples

Some examples include:
ClassSubclassesActivators
Calcium-activated
6T & 1P

  • 1-EBIO
  • NS309
  • CyPPABKCa-specific:
  • * Flufenamic acid
  • * Meclofenamic acid
  • * Niflumic acid
  • * Nimesulide
  • * Rottlerin (mallotoxin)
  • * Tolfenamic acid
  • Inwardly rectifying 2T & 1P
  • none
  • Inwardly rectifying 2T & 1P
  • GPCR agonists
  • ML-297 (VU0456810)
  • Inwardly rectifying 2T & 1P
  • Aprikalim
  • Bimakalim
  • Cromakalim
  • Diazoxide
  • Emakalim
  • Levcromakalim
  • Mazokalim
  • Minoxidil
  • Naminidil
  • Nicorandil
  • Pinacidil
  • Rilmakalim
  • Sarakalim
  • Tandem pore domain 4T & 2P
  • halothane
  • Riluzole
  • Arachidonic acid
  • Voltage-gated 6T & 1P
    KCNQ (Kv7)-specific:
  • Flupirtine
  • Retigabine
  • XEN1101