Plakohypaphorine


Plakohypaphorines are halogenated indolic non-proteinogenic amino acids named for their similarity to hypaphorine. First reported in the Caribbean sponge Plakortis simplex in 2003, plakohypaphorines A-C were the first iodine-containing indole alkaloids to be discovered in nature. Plakohypaphorines D-F, also found in P. simplex, were reported in 2004 by a group including the researchers who discovered the original plakohypaphorines.
PlakohypaphorineChemical nameChemical formulaSMILESImage
Plakohypaphorine7-Iodo-N,N,N-trimethyltryptophanC14H17IN2O2OCCCc2cnc1c2cccc1I
Plakohypaphorine B6,7-Diiodo-N,N,N-trimethyltryptophanC14H16I2N2O2OCCCc2cnc1c2cccc1I
Plakohypaphorine C5,7-Diiodo-N,N,N-trimethyltryptophanC14H16I2N2O2CNCCc2cnc1c2cccc1I
Plakohypaphorine D5,6-Diiodo-N,N,N-trimethyltryptophanC14H16I2N2O2Ic2cc1cncc1CCNC
Plakohypaphorine E5,6,7-Triiodo-N,N,N-trimethyltryptophanC14H15I3N2O2CNCCc1cncc1cc2I
Plakohypaphorine F6-Chloro-5-iodo-N,N,N-trimethyltryptophanC14H16ClIN2O2Clc2c1nccc1ccc2